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Name: 2',5'-Dimethoxyfentanyl (N-(1-(2,5-dimethoxyphenethyl)piperidin-4-yl)-N-phenylpropionamide)
Type: Opioid derivative
AKA: N/A
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II. Natural Derivative
Synthetic substance, no natural derivative
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III. Chemical Profile (IUPAC name)
2',5'-Dimethoxyfentanyl (N-(1-(2,5-dimethoxyphenethyl)piperidin-4-yl)-N-phenylpropionamide)
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IV. History
2',5'-Dimethoxyfentanyl is a synthetic opioid and analog of fentanyl. It has been identified in the illicit drug market and is known for its high potency and risk of overdose. The emergence of such synthetic opioids underscores the ongoing challenges in controlling their production and distribution, contributing to the opioid epidemic.
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V. Legal Information
2',5'-Dimethoxyfentanyl, a potent synthetic opioid, is regulated as a controlled substance in many countries due to its high potential for abuse. In the US, it is covered under the Federal Analog Act if considered similar to fentanyl. Globally, it faces strict regulations reflecting concerns about opioid addiction and misuse.
US Federal Schedule - I
Schedule I drugs, substances, or chemicals are defined as drugs with no currently accepted medical use and a high potential for abuse. Some examples of Schedule I drugs are: heroin, lysergic acid diethylamide (LSD), marijuana (cannabis), 3,4-methylenedioxymethamphetamine (ecstasy), methaqualone, and peyote.
Key US Federal Policies:
Controlled Substances Act. Public Law: Public Law 91-513 (text can be found on GovInfo) (https://www.dea.gov/drug-information/csa). Date enacted: October 27, 1970.
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VI. Physical Effects
2',5'-Dimethoxyfentanyl, a potent synthetic opioid, provides significant analgesia. As a downer, it induces sedation and respiratory depression. Short-term effects include pain relief and euphoria, while long-term use can lead to addiction and tolerance. Overdose risks involve severe respiratory issues and potential fatality. Safe dosing requires careful medical supervision. Recent findings focus on its potency and the associated risks of addiction and overdose.  |
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VII. Psychological Effects
2',5'-Dimethoxyfentanyl, a potent synthetic opioid, impacts opioid receptors to produce intense euphoria and sedation. Psychological effects include mood swings and cognitive impairment. Immediate effects last several hours, with long-term use leading to dependence and severe mental health issues. Research examines its potency, abuse potential, and safety.
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VIII. Culture
2',5'-Dimethoxyfentanyl is a synthetic opioid with no historical or cultural lore, emerging in recent years. Its cultural significance is tied to discussions about synthetic opioids, their regulation, and their impact on public health. Proponents of strict regulation highlight its potential for abuse and overdose, while some argue for its controlled medical use. Its primary impact is seen in the context of the opioid epidemic, reflecting broader societal challenges in managing synthetic opioid proliferation.
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