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Name: 4-Methylaminorex (cis isomer)
Type: Stimulant
AKA: U4Euh, McN-422
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II. Natural Derivative
Synthetic substance, no natural derivative
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III. Chemical Profile (IUPAC name)
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IV. History
4-Methylaminorex, a synthetic stimulant, was first synthesized in the 1970s. The cis isomer of this compound was developed to study its stimulant properties. Known for its potent effects, 4-methylaminorex gained popularity in the illicit drug market as a 'designer drug' due to its stimulant effects. Its emergence highlighted the challenges of controlling synthetic stimulants and managing their potential for abuse and health risks. Regulatory actions have been implemented to address its use and mitigate associated health concerns.
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V. Legal Information
4-Methylaminorex, a stimulant, is classified as a Schedule I controlled substance in the US, making it illegal. Many countries have similarly banned it due to its potent stimulant effects and health risks. The UNODC monitors new psychoactive substances, emphasizing the need for international regulation to prevent misuse. Trends show increasing control measures to address the growing issue of synthetic drug use.
US Federal Schedule - I
Schedule I drugs, substances, or chemicals are defined as drugs with no currently accepted medical use and a high potential for abuse. Some examples of Schedule I drugs are: heroin, lysergic acid diethylamide (LSD), marijuana (cannabis), 3,4-methylenedioxymethamphetamine (ecstasy), methaqualone, and peyote.
Key US Federal Policies:
Controlled Substances Act. Public Law: Public Law 91-513 (text can be found on GovInfo) (https://www.dea.gov/drug-information/csa). Date enacted: October 27, 1970.
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VI. Physical Effects
4-Methylaminorex (cis isomer) is a stimulant with effects similar to amphetamines. It acts as an upper, increasing energy and alertness. Short-term use can lead to euphoria and heightened physical performance, but long-term use poses risks of cardiovascular issues and psychological effects. Overdose risks include severe agitation and cardiovascular effects. Safe use requires cautious dosing. Recent research explores its stimulant effects and health risks.  |
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VII. Psychological Effects
4-Methylaminorex, a stimulant, affects monoamine neurotransmitters, causing increased alertness and euphoria. Immediate effects include mood enhancement and cognitive stimulation, lasting several hours. Long-term use can lead to dependence, anxiety, and cognitive decline. Research indicates significant mental health risks with chronic use, including severe anxiety and potential for psychosis.
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VIII. Culture
4-Methylaminorex is a stimulant with effects similar to amphetamines. Its cultural significance lies in its use as a recreational drug and its potential for abuse. Media coverage often addresses its stimulant properties and the risks associated with its use. 4-Methylaminorex is used recreationally rather than medicinally and contributes to discussions about stimulant use and drug regulation.
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