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Name: Alphacetylmethadol except levo-alphacetylmethadol
Type: Opioid analgesic
AKA: N/A
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II. Natural Derivative
Synthetic substance, no natural derivative
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III. Chemical Profile (IUPAC name)
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IV. History
Alpha-Acetylmethadol, a synthetic opioid, was developed in the mid-20th century. It is used for pain management and addiction treatment. Its history reflects its role in opioid research and the challenges of managing its abuse potential.
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V. Legal Information
Alphaacetylmethadol is an opioid with abuse potential. It is controlled to prevent misuse and addiction, with global regulation reflecting concerns about its effects. [Source: UNODC].
US Federal Schedule - I
Schedule I drugs, substances, or chemicals are defined as drugs with no currently accepted medical use and a high potential for abuse. Some examples of Schedule I drugs are: heroin, lysergic acid diethylamide (LSD), marijuana (cannabis), 3,4-methylenedioxymethamphetamine (ecstasy), methaqualone, and peyote.
Key US Federal Policies:
Controlled Substances Act. Public Law: Public Law 91-513 (text can be found on GovInfo) (https://www.dea.gov/drug-information/csa). Date enacted: October 27, 1970.
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VI. Physical Effects
Alphacetylmethadol, except levo-alphacetylmethadol, is an opioid used for pain relief. It causes sedation, respiratory depression, and constricted pupils. Short-term use provides effective pain management, while long-term use can lead to addiction and respiratory issues. Overdose risks include severe respiratory depression and potential death. Safe use requires medical supervision. Recent research emphasizes its potency and associated risks with opioid use.  |
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VII. Psychological Effects
Alpha-acetylmethadol (except levo-alpha-acetylmethadol) is an opioid with effects on mu-opioid receptors, leading to euphoria and sedation. Immediate effects include mood enhancement and pain relief, lasting several hours. Long-term use may result in addiction, cognitive impairments, and mood disturbances. Research emphasizes its potential for dependence and impact on opioid receptor systems.
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VIII. Culture
Alpha-acetylmethadol (except levo-alpha-acetylmethadol) is an opioid used for pain relief and as a methadone alternative, classifying it as a downer. Short-term use provides effective analgesia, while long-term use can lead to dependence, tolerance, and severe health issues. Overdose risks include severe respiratory depression and potentially fatal outcomes. Safe dosages are typically prescribed and controlled by medical professionals. Recent research highlights its effectiveness in pain management but warns of high abuse potential. Physical effects include drowsiness, constricted pupils, and respiratory depression.
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