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Name: Anileridine
Type: Opioid analgesic
AKA: Leritine
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II. Natural Derivative
Synthetic substance, no natural derivative
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III. Chemical Profile (IUPAC name)
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IV. History
Anileridine, an opioid analgesic, was developed in the 20th century. It is used for pain management and is part of the broader category of opioids used in medical treatments.
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V. Legal Information
Anileridine is an opioid analgesic with potential for abuse. It is regulated in the United States as a Schedule II controlled substance and similarly controlled in other countries to manage its use and prevent misuse. [Source: UNODC].
US Federal Schedule - II
Schedule II drugs, substances, or chemicals are defined as drugs with a high potential for abuse, with use potentially leading to severe psychological or physical dependence. These drugs are also considered dangerous. Some examples of Schedule II drugs are: combination products with less than 15 milligrams of hydrocodone per dosage unit (Vicodin), cocaine, methamphetamine, methadone, hydromorphone (Dilaudid), meperidine (Demerol), oxycodone (OxyContin), fentanyl, Dexedrine, Adderall, and Ritalin.
Key US Federal Policies:
Controlled Substances Act. Public Law: Public Law 91-513 (text can be found on GovInfo) (https://www.dea.gov/drug-information/csa). Date enacted: October 27, 1970.
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VI. Physical Effects
Anileridine is a synthetic opioid with analgesic effects. It causes sedation, respiratory depression, and constricted pupils. Short-term use is effective for pain management, but long-term use can lead to addiction, tolerance, and severe health issues. Overdose risks include fatal respiratory depression. Safe use involves strict dosing and medical supervision. Recent research explores its efficacy and safety profile compared to other opioids.  |
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VII. Psychological Effects
Anileridine, an opioid analgesic, affects mu-opioid receptors, producing euphoria and sedation. Immediate effects include pain relief and mood elevation, lasting several hours. Long-term use may lead to addiction, cognitive impairments, and mood disturbances. Research highlights its efficacy as an analgesic and associated risks of psychological dependence and cognitive effects.
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VIII. Culture
Anileridine is an opioid analgesic providing pain relief, classifying it as a downer. Short-term use alleviates severe pain, while long-term use can lead to dependence and tolerance. Overdose is highly possible, causing respiratory depression and potentially fatal outcomes. Safe dosages are medically prescribed, typically under 100 mg per day. Recent research highlights its efficacy in pain management but warns of addiction risks. Physical effects include drowsiness, constricted pupils, and respiratory depression.
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