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Name: Cenobamate [(1R)-1-(2-chlorophenyl)-2-(tetrazol-2-yl)ethyl]carbamate
Type: Anticonvulsant
AKA: 2H-tetrazole-2-ethanol, alpha-(2-chlorophenyl)-, carbamate (ester), (alphaR)-; carbamic acid (R)-(+)-1-(2-chlorophenyl)-2-(2H-tetrazol-2-yl)ethyl ester)
![Cenobamate [(1R)-1-(2-chlorophenyl)-2-(tetrazol-2-yl)ethyl]carbamate image](https://grammasearch.com/dev/v2/aiimages/cenobamate_%5B%281r%29-1-%282-chlorophenyl%29-2-%28tetrazol-2-yl%29ethyl%5Dcarbamate.png)
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II. Natural Derivative
Synthetic substance, no natural derivative
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III. Chemical Profile (IUPAC name)
![Cenobamate [(1R)-1-(2-chlorophenyl)-2-(tetrazol-2-yl)ethyl]carbamate image](/dev/v2/pages/pubchem_images/124081426.png)
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IV. History
Cenobamate, an anticonvulsant, was developed in the 2010s for the treatment of epilepsy. Its development reflects ongoing research into effective treatments for neurological disorders. Cenobamate's introduction has provided a new option for managing seizures with a focus on efficacy and safety.
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V. Legal Information
Cenobamate is an anticonvulsant used for epilepsy. It is classified as a Schedule V controlled substance in the U.S. due to its potential for abuse. Globally, its regulation is aligned with efforts to manage its use and prevent misuse. [Source: UNODC].
US Federal Schedule - V
Schedule V drugs, substances, or chemicals are defined as drugs with lower potential for abuse than Schedule IV and consist of preparations containing limited quantities of certain narcotics. Schedule V drugs are generally used for antidiarrheal, antitussive, and analgesic purposes. Some examples of Schedule V drugs are: cough preparations with less than 200 milligrams of codeine or per 100 milliliters (Robitussin AC), Lomotil, Motofen, Lyrica, Parepectolin.
Key US Federal Policies:
Controlled Substances Act. Public Law: Public Law 91-513 (text can be found on GovInfo) (https://www.dea.gov/drug-information/csa). Date enacted: October 27, 1970.
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VI. Physical Effects
Cenobamate is a medication used to treat seizures. It has sedative effects and modulates brain activity, acting as a downer. Short-term use helps control seizures, while long-term use is generally safe with monitored dosing. Overdose risks include excessive sedation and respiratory depression. Safe use involves following prescribed dosages and regular medical supervision. Recent research highlights its efficacy in treating refractory seizures and its safety profile.  |
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VII. Psychological Effects
Cenobamate is an anticonvulsant used for seizure disorders, improving mood and reducing anxiety. Long-term use is generally well-tolerated, though research is ongoing to understand its full psychological impact and risks.
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VIII. Culture
Cenobamate is a medication used to treat epilepsy, classifying it as a downer. Short-term use reduces seizure frequency and improves control, while long-term use can lead to cognitive impairment and dependence. Overdose risks include severe sedation and potential respiratory depression. Safe dosages are typically prescribed by medical professionals. Recent research highlights its efficacy in managing epilepsy but notes potential side effects such as sedation and cognitive effects. Physical effects include reduced seizure activity, drowsiness, and potential for respiratory depression.
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