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Name: Furethidine
Type: Antihypertensive
AKA: N/A
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II. Natural Derivative
Synthetic substance, no natural derivative
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III. Chemical Profile (IUPAC name)
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IV. History
Furethidine, an opioid analgesic, was developed in the 20th century. It was used for pain management but has been largely replaced by newer medications due to safety concerns and the development of more effective pain relievers.
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V. Legal Information
Furethidine, an opioid analgesic, is classified as a Schedule I substance in the US, making it illegal. Its high potential for abuse and lack of accepted medical use lead to similar bans in many countries. The UNODC and other regulatory bodies emphasize strict control measures to prevent misuse and address the opioid crisis.
US Federal Schedule - I
Schedule I drugs, substances, or chemicals are defined as drugs with no currently accepted medical use and a high potential for abuse. Some examples of Schedule I drugs are: heroin, lysergic acid diethylamide (LSD), marijuana (cannabis), 3,4-methylenedioxymethamphetamine (ecstasy), methaqualone, and peyote.
Key US Federal Policies:
Controlled Substances Act. Public Law: Public Law 91-513 (text can be found on GovInfo) (https://www.dea.gov/drug-information/csa). Date enacted: October 27, 1970.
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VI. Physical Effects
Furethidine is a synthetic opioid used for pain relief. It acts as a downer, causing sedation, respiratory depression, and constricted pupils. Short-term use provides pain relief, but long-term use may lead to addiction, tolerance, and severe health issues. Overdose risks include fatal respiratory depression. Safe use requires strict dosing and medical oversight. Recent research highlights its potency and risks associated with prolonged use.  |
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VII. Psychological Effects
Furethidine, an opioid analgesic, affects mu-opioid receptors, providing mood enhancement and pain relief. Immediate effects include euphoria and sedation, lasting several hours. Long-term use can lead to dependence, cognitive impairments, and mood disturbances. Research highlights the risks of psychological dependence and cognitive decline with chronic use.
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VIII. Culture
Furethidine, an opioid analgesic, provides pain relief and sedation, classifying it as a downer. Short-term use alleviates severe pain, while long-term use can lead to dependence and tolerance. Overdose is highly possible, causing respiratory depression and potentially fatal outcomes. Safe dosages are strictly prescribed, typically under 100 mg per day. Recent research stresses the need for cautious prescribing to avoid addiction. Physical effects include drowsiness, constricted pupils, and reduced pain sensation.
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