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Name: Isovaleryl fentanyl (3-methyl-N-(1-phenethylpiperidin-4-yl)-N-phenylbutanamide)
Type: Synthetic opioid
AKA: N/A
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II. Natural Derivative
Synthetic substance, no natural derivative
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III. Chemical Profile (IUPAC name)
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IV. History
Isovaleryl Fentanyl, a synthetic opioid, was developed in the early 21st century. It is used in research to explore its effects on opioid receptors. Its development reflects the ongoing innovation in synthetic opioids and their implications for pain management and drug policy.
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V. Legal Information
Isovaleryl fentanyl is a potent synthetic opioid, classified under strict controls due to its high potential for abuse. In the U.S., it is regulated under the Federal Analog Act, which covers substances similar to fentanyl. Internationally, its legal status reflects increased regulation to manage the risks associated with synthetic opioids. [Source: UNODC].
US Federal Schedule - I
Schedule I drugs, substances, or chemicals are defined as drugs with no currently accepted medical use and a high potential for abuse. Some examples of Schedule I drugs are: heroin, lysergic acid diethylamide (LSD), marijuana (cannabis), 3,4-methylenedioxymethamphetamine (ecstasy), methaqualone, and peyote.
Key US Federal Policies:
Controlled Substances Act. Public Law: Public Law 91-513 (text can be found on GovInfo) (https://www.dea.gov/drug-information/csa). Date enacted: October 27, 1970.
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VI. Physical Effects
Isovaleryl fentanyl is a synthetic opioid with strong analgesic effects. It acts as a downer, causing sedation and respiratory depression. Short-term use is effective for pain management, but long-term use can lead to addiction, tolerance, and severe health issues. Overdose risks include fatal respiratory depression. Safe use requires strict dosing and medical supervision. Recent research explores its efficacy and risks compared to other opioids.  |
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VII. Psychological Effects
Isovaleryl fentanyl is a potent synthetic opioid providing euphoria, sedation, and analgesia. Immediate effects include mood elevation and cognitive impairment. Long-term use can lead to dependence, tolerance, and severe withdrawal symptoms. Chronic use is associated with mood disorders, cognitive decline, and high overdose risk. Recent research underscores its potency and high abuse potential, similar to other potent opioids.
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VIII. Culture
Isovaleryl fentanyl is a synthetic opioid with no significant historical or cultural lore. It is part of the broader opioid crisis, with recreational use leading to significant health risks and societal issues. Its modern cultural impact is tied to the debates over synthetic opioids, their regulation, and their role in the opioid epidemic. Proponents of strict regulation emphasize the dangers of abuse and overdose, while some argue for its medical utility under controlled conditions. Its use is primarily illicit, contributing to public health and law enforcement challenges.
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