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Name: N-pyrrolidino etonitazene; etonitazepyne (2-(4-ethoxybenzyl)-5-nitro-1-(2- (pyrrolidin-1-yl)ethyl)-1H-benzimidazole)
Type: Opioid
AKA: 2-(4-ethoxybenzyl)-5-nitro-1-(2-(pyrrolidin-1-yl)ethyl)-1H-benzimidazole, Synthetic Opioids
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II. Natural Derivative
Synthetic substance, no natural derivative
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III. Chemical Profile (IUPAC name)
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IV. History
N-Pyrrolidino etonitazene, also known as etonitazepyne, is a synthetic opioid and part of the benzimidazole class of opioids. It has been identified in the illicit drug market and is known for its high potency and risk of overdose. The development and distribution of such synthetic opioids pose significant challenges to public health and law enforcement.
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V. Legal Information
N-Pyrrolidino-etonitazene, a synthetic opioid, is regulated as a controlled substance due to its high potential for abuse. In the US, it is classified under analog laws similar to fentanyl. Globally, its legal status is increasingly restrictive, reflecting efforts to manage synthetic opioids and prevent misuse.
US Federal Schedule - I
Schedule I drugs, substances, or chemicals are defined as drugs with no currently accepted medical use and a high potential for abuse. Some examples of Schedule I drugs are: heroin, lysergic acid diethylamide (LSD), marijuana (cannabis), 3,4-methylenedioxymethamphetamine (ecstasy), methaqualone, and peyote.
Key US Federal Policies:
Controlled Substances Act. Public Law: Public Law 91-513 (text can be found on GovInfo) (https://www.dea.gov/drug-information/csa). Date enacted: October 27, 1970.
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VI. Physical Effects
N-Pyrrolidino Etonitazene and Etonitazepyne, synthetic opioids, provide significant analgesia. As downers, they cause sedation and respiratory depression. Short-term effects include pain relief and euphoria, while long-term use can lead to addiction and tolerance. Overdose risks involve severe respiratory issues and potential fatality. Safe dosing requires careful medical supervision. Recent research highlights their potency and the need for cautious use to avoid addiction.  |
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VII. Psychological Effects
N-Pyrrolidino Etonitazene, a potent opioid, interacts with opioid receptors to produce strong euphoria and pain relief. Psychological effects include mood alteration and cognitive impairment. Immediate effects last several hours, with risks of severe dependence and mental health issues with long-term use. Research focuses on its potency, safety, and potential for abuse.
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VIII. Culture
N-Pyrrolidino Etonitazene, a synthetic opioid, has no historical or cultural lore, being a recent development. It is part of the broader opioid crisis, with significant health risks and societal issues related to its use. Its modern cultural impact is tied to debates over synthetic opioids, their regulation, and their role in the opioid epidemic. Proponents of strict regulation emphasize the dangers of abuse and overdose, while some argue for its medical utility under controlled conditions. Its use is primarily illicit, contributing to public health and law enforcement challenges.
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